IntroPharmaI Drugs
Terms
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CHOLOMIMETICS:
direct-acting (receptor agonists)
choline esters: -
Ach (Miochol)
bethanechol (Urecholin)
carbachol (Miostat)
methacholine -
CHOLOMIMETICS:
direct-acting (receptor agonists)
alkaloids -
muscarine (M)
pilocarpine (M, Pilocar)
nicotine (N) -
CHOLOMIMETICS:
indirect-acting (anti-cholinesterases)
- reversible
- carbamates -
edrophonium (Tensilon)
demecarium (Humorsol)
neostigine (Prostigmin)
physostigmine (generic)
pyridostigmine (Mestinon) -
CHOLOMIMETICS:
indirect-acting (anti-cholinesterases)
- reversible
- for Alzheimers disease -
donepezil (Aricept)
galntamine (Reminyl) -
CHOLOMIMETICS:
indirect-acting (anti-cholinesterases)
- irreversible
- organophosphates -
echothiophate (phosholine)
malathion
parathion
soman -
CHOLOMIMETICS:
acute narrow angle glaucoma
- muscarinic agonist -
pilocarpine (Pilocar) drops
carbachol (Isopto-carbachol) drops -
CHOLOMIMETICS:
acute narrow angle glaucoma
anticholinesterase -
- physostigmine ophth. ointment
- echothiophate (Phospholine) drops
- demecarium (Humorsol) drops -
CHOLOMIMETICS:
chronic open angle glaucoma
anticholinesterase - - physostigmine
-
CHOLOMIMETICS:
chronic open angle glaucoma
muscarinic agonist -
- pilocarpine
- carbachol -
Non-CHOLOMIMETICS:
chronic open angle glaucoma
carbonic anhydrase inhibitors -
- acetazolamide (Diamox)
- brinzolamide (Azopt) -
Non-CHOLOMIMETICS:
chronic open angle glaucoma
prostaglandins -
- bimatoprost (lumigan)
- unoprostone (Rescula) -
Non-CHOLOMIMETICS:
chronic open angle glaucoma
alpha agonists - non-selective -
- epinephrine
- dipivefrin (Propine) -
Non-CHOLOMIMETICS:
chronic open angle glaucoma
alpha-2 agonists -
- aproclonidine (Iopidine)
- brimonidine (Alphagan) -
Non-CHOLOMIMETICS:
chronic open angle glaucoma
beta blockers -
- betaxolol ( Betoptic )
- timolol ( Timoptic, Betimol) -
CHOLOMIMETICS:
GI and urinary tract
anticholinesterase - neostigmine (Prostigmin)
-
CHOLOMIMETICS:
GI and urinary tract
muscarinic agonist - bethanechol (Urecholine)
-
CHOLOMIMETICS:
GI and urinary tract
for GERD - H2 blockers
-
CHOLOMIMETICS:
dry mouth
muscarinic agonist - cevimiline (Evoxac)
-
CHOLOMIMETICS:
Myasthenia Gravis (MG)
anticholinesterase for diagnosis - - edrophonium (Tensilon )
-
CHOLOMIMETICS:
Myasthenia Gravis (MG)
anticholinesterase to assess level of long term treatment - - edrophonium (Tensilon )
-
CHOLOMIMETICS:
Myasthenia Gravis (MG)
anticholinesterase long term treatment -
- pyridostigmine ( Mestinon )
- neostigmine (Prostigmin )
- ambenonium (Mytelase )
- demercarium ( Humorsol ) -
CHOLOMIMETICS:
reversal of surgical neuromuscular blockade
anticholinesterase -
- neostigmine (Prostigmin )
- pyridostigmine ( Mestinon )
- edrophonium (Tensilon ) -
CHOLOMIMETICS:
reversal of surgical neuromuscular blockade
depolarizing drugs - - succinylcholine
-
CHOLOMIMETICS:
reversal of surgical neuromuscular blockade
non-polarizing drugs -
- curare
- atracurium
- pipecuronium
- pancuronium
- vecuronium -
CHOLOMIMETICS:
antidote for insecticides and humanocides - - atropine (Protopam, 2-PAM)
-
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
prototype - - atropine (Protopam, 2-PAM)
-
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
synthetic tertiary ammonium analogues of atropine -
- dicyclomine (Bentyl)
- tropicamide (Mydriacil) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
synthetic tertiary ammonium analogues of atropine
antihistamines -
- dimenhydrinate (Dramamine)
- diphenhydramine (Benadryl) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
synthetic tertiary ammonium analogues of atropine
tricyclic antidepressants - - amitriptyline (Elavil)
-
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
synthetic tertiary ammonium analogues of atropine
antipsychotics -
- haloperidol (Haldol)
- chlorpromazine (Thorazine) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
for fundoscopic exam -
- tropicamide (Mydriacil)
- cyclopentolate (Cyclogil)
- Atropine sulfate (Isopto Atropine) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
for IBS and peptic ulcer -
- glycopyrrolate (Robinul) 4o
- dicyclomine (Bentyl) 3o
- hyoscyamine (Levsin) 3o
- hyoscyamine + phenobarbital (Donnatal) 3o
- clidinium + chlordiazepoxide (Librax) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
for traveler's diarrhea & other mild GI tract hypomotility - atropine + diphenoxylate (Lomotil)
-
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
NO antimuscarinic agents, just opioid
for traveler's diarrhea & other mild GI tract hypomotility -
- loperamide (Imodium A-D) OTC
- loperamide (Imodium) Rx -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
for overactive bladder and urge incontinence -
- oxybutynin (Ditropan)
- tolterodine (Detrol LA) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
as adjunct to surgical anesthesia -
- no longer used
- replaced by halothane, enflurane or isoflurane -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
for asthma & COPD -
- ipratropium (Atrovent)
- tiotropium (Spiriva)
- ipratropium + albuterol (Combivent) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
adjunct for Parkinson's Disease -
- benztropine (Cogentin)
- trihexyphenidyl (Artane)
- diphenhydramine (Benadryl inj.) -
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
antimuscarinic agents
(Muscarinic Receptor Blockers)
for motion sickness - scopolamine (Transderm Scop)- a dermal patch
-
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics)
Non - antimuscarinic agent
(Muscarinic Receptor Blockers)
antihistamines for motion sickness with antimuscarinic effects -
- dimenhydrinate (Dramamine)
- meclizine (Antivert) - for poisoning from cholinomimetic agent
- - atropine
- Antidotes for insecticides and humanocides
-
- atropine (Isopto Atropine)
- pralidoxime (Protopam, 2-PAM)