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Pharmacology second test

Terms

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Tetrodotoxin
Sodium Channel Inhibitors
Saxotoxin
Sodium Channel Inhibitors
Procaine
Sodium Channel Inhibitors
Hemicholinium-3
ACh synthesis/release - choline
Vesamicol
ACh synthesis/release - storage
Botulinum
ACh synthesis/release
Latrotoxin
ACh synthesis/release
Edrophonium
ACh esterase inhibitors - reversible competitive, diagnose MG
Tacrine
ACh esterase inhibitors - reversible competitive
Neostigmine
ACh esterase inhibitors - carbamate ester
Physostigmine
ACh esterase inhibitors - carbamate ester
DFP
ACh esterase inhibitors - organophosphate, chemical weapon
Malathion/Parathion
ACh esterase inhibitors - organophosphate, insecticide
Soman
ACh esterase inhibitors - organophosphate, nerve gas
Pralidoxime
2-PAM - reactivates AChE
Methacholine
Muscarinic receptor agonists - M2
Bethanechol
Muscarinic receptor agonists - primarily for smooth muscle
Pilocarpine
Muscarinic receptor agonists - glaucoma
Muscarine
Muscarinic receptor agonists
McN-A343
Muscarinic receptor agonists - M1
Atropine
Muscarinic receptor antagonists
Scopolamine
Muscarinic receptor antagonists
Pirenzepine
Muscarinic receptor antagonists - M1
Ipratropium
Muscarinic receptor antagonists
Propantheline
Muscarinic receptor antagonists
Tropicamide
Muscarinic receptor antagonists - used in the eye
Tolterodine
Muscarinic receptor antagonists - used for overactive bladder
Nicotine
Nicotinic receptor agonists
Succinylcholine
Nicotinic receptor agonists
Decamethonium
Nicotinic receptor agonists
Tubocurarine
Nicotinic receptor antagonists
Pipecuronium
Nicotinic receptor antagonists - long duration
Pancuronium
Nicotinic receptor antagonists - intermediate duration
Vecuronium
Nicotinic receptor antagonists - intermediate duration
Mivacurium
Nicotinic receptor antagonists - short duration
Hexamethonium
Nicotinic receptor antagonists
Mecamylamine
Nicotinic receptor antagonists
Resperipine
Indirect acting adrenergic agents - destroys vesicles containing NT
Guanethidine
Indirect acting adrenergic agents - taken up by uptake 1 and displaces NE
Metyrosine
Catecholamine sythesis/metabolism - interrupts tyrosine hydroxylase
MAO inhibitors
Catecholamine sythesis/metabolism - prevents breakdown of NT
COMT inhibitors
Catecholamine sythesis/metabolism - synthesis of NT
Methyldopa
Catecholamine sythesis/metabolism - false transmitter
Cocaine
Catecholamine sythesis/metabolism
Amphetamines
Catecholamine sythesis/metabolism
Tricyclic antidepressants
Catecholamine sythesis/metabolism
Phenylephrine
Adrenergic receptor agonists - alpha 1
Oxymetolazine
Adrenergic receptor agonists - alpha 1
Clonidine
Adrenergic receptor agonists - alpha 2
Brimonidine
Adrenergic receptor agonists - alpha 2
Phenoxybenzamine
Adrenergic receptor antagonists - alpha irreversible
Prazosin
Adrenergic receptor antagonists - alpha 1
Tamsulosin
Adrenergic receptor antagonists - alpha 1
Yohimbine
Adrenergic receptor antagonists - alpha 2
Isoproterenol
Beta receptor agonists
Dobutamine
Beta receptor agonists - beta 1
Metaproterenol
Beta receptor agonists - beta 2
Salmeterol
Beta receptor agonists
Albuterol
Beta receptor agonists
Bitolterol
Beta receptor agonists
Propanolol
Beta receptor antagonists - nonselective
Nadolol
Beta receptor antagonists - nonselective
Pindolol
Beta receptor antagonists - nonselective
Timolol
Beta receptor antagonists - nonselective
Labetolol
Beta receptor antagonists - nonselective
Esmolol
Beta receptor antagonists - beta 1
Atenolol
Beta receptor antagonists - beta 1
Metoprolol
Beta receptor antagonists - beta 1
Carteolol
Beta receptor antagonists - 3rd generation
Carvedilol
Beta receptor antagonists - 3rd generation

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